GP 2a

Name: GP 2a
Brand: Tocris Bioscience
SKU: 2678
Price: 199 USD

Catalog #: 2678 Datasheet / COA / SDS

Discontinued Product

2678 has been discontinued.

View all Cannabinoid R2/CB2 Agonists products.

GP 2a | CAS No. 919077-81-9 | Cannabinoid R2/CB2 Agonists

1 Image

Description: Selective CB2 agonist

Chemical Name: N-Cyclohexyl-1-(2,4-dichlorophenyl)-1,4-dihydro-6-methylindeno[1,2-c]pyrazole-3-carboxamide

Purity: ≥99%

View All Products for Cannabinoid R2/CB2 Agonists

Product Details

Reviews

Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

GP 2a is a selective CB₂ receptor agonist; K_i values are 7.6 and 900 nM for CB₂ and CB₁ receptors respectively. Increases P-ERK1/2 expression in HL-60 cells in vitro.

Technical Data

M.Wt:

440.36

Formula:

C₂₄H₂₃Cl₂N₃O

Solubility:

Soluble to 50 mM in DMSO and to 20 mM in ethanol

Purity:

≥99%

Storage:

Store at RT

CAS No:

919077-81-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxam
Murineddu et al.
J.Med.Chem., 2006;49:7502

Product Datasheets

COA view current batch

SDS

Reconstitution Calculator

Molarity Calculator

Reconstitution Calculator

Molarity Calculator

Mass

Concentration

Volume

M. Wt* g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

Reviews for GP 2a

There are currently no reviews for this product. Be the first to review GP 2a and earn rewards!

Have you used GP 2a?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review

Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.