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GSK 2879552

Catalog #: 8128 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
8128/10
8128/50

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GSK 2879552 | CAS No. 1902123-72-1 | Histone Demethylase Inhibitors
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Description: Lysine-Specific Demethylase 1 (LSD1) inhibitor

Chemical Name: 4-[[4-[[[(1R,2S)-2-Phenylcyclopropyl]amino]methyl]-1-piperidinyl]methyl]benzoic acid dihydrochloride

Purity: ≥98%

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Biological Activity

GSK 2879552 is a selective lysine-specific demethylase 1 (LSD1) inhibitor. When combined with other small molecules (EPZ-5676, N-methyl-d-aspartate and Bay K 8644), GSK 2879552 accelerates maturation of human pluripotent stem cell-derived neurons. GSK 2879552 inhibits the growth of small cell lung carcinoma (SCLC) and AML lines. In vivo, GSK 2879552 (1.5 mg/kg, p.o.) demonstrates tumor growth inhibition in SCLC xenograph mouse models.

Technical Data

M.Wt:
437.41
Formula:
C23H28N2O2.2HCl
Solubility:
Soluble to 50 mM in DMSO and to 20 mM in water
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1902123-72-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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