Iodophenpropit dihydrobromide

Key Product Details

Product Description

Iodophenpropit dihydrobromide is a selective H₃ antagonist with high affinity (K_D = 0.3 nM).

Licensing Information

Sold with the permission of SCI, Amsterdam

Product Specifications for Iodophenpropit dihydrobromide

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for Iodophenpropit dihydrobromide

The following data is based on the product molecular weight 576.13.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

2 Recalculate

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.25 mM	6.94 mL	34.71 mL	69.43 mL
1.25 mM	1.39 mL	6.94 mL	13.89 mL
2.5 mM	0.69 mL	3.47 mL	6.94 mL
12.5 mM	0.14 mL	0.69 mL	1.39 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 11 publications citing the usage of this product.

• Shahid Histamine, histamine receptors, and their role in immunomodulation: An updated systematic review. Open Immunol.J.
• Jansen Characterisation of the binding of the first selective radiolabelled histamine H₃ receptor antagonist, [¹²⁵I]-iodophenpropit, to rat brain. Br.J.Pharmacol. 1994 PMID: 7834183
• Menge Synthesis of S-[3-(4(5)-imidazolyl)propyl]-N-[2-(4-[¹²⁵I]-iodophenylethyl]isothiourea sulfate [¹²⁵I]-iodophenpropit), a new probe for histamine H₃ receptor binding sites. J.Labelled Comp.Radiopharm. XXXI
• Jansen The first radiolabelled histamine H₃ receptor antagonist, [¹²⁵I]iodophenpropit: saturable and reversible binding to rat cortex membranes. Eur.J.Pharmacol. 1992 PMID: 1330590

Product Documents for Iodophenpropit dihydrobromide