Lenalidomide 5'-piperazine-4-methylpiperidine

Tocris Bioscience | Catalog # 7473

Cereblon ligand with terminal piperidine for onward chemistry
Tocris Bioscience

Key Product Details

Description

Cereblon ligand with terminal piperidine for onward chemistry
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Product Description

Lenalidomide 5'-piperazine-4-methylpiperidine is a functionalized cereblon ligand for PROTAC® research and development; incorporates an E3 ligase ligand with a terminal piperidine for onward chemistry to generate Protein Degraders with rigid linkers. Part of a range of functionalized tool molecules for PROTAC R&D.

Please contact us for SD files of our available Degrader Building Blocks.

PROTAC® is a registered trademark of Arvinas Operations, Inc., and is used under license.

Usage Guidelines

This product is provided for use in onward chemistry. Suitable solvents can be used.

Product Specifications for Lenalidomide 5'-piperazine-4-methylpiperidine

Molecular Weight

498.45

Formula

C23H31N5O3.2HCl

Storage

Store at -20°C

Purity

≥94% (HPLC)

Chemical Name

3-[1,3-Dihydro-1-oxo-5-[4-(4-piperidinylmethyl)-1-piperazinyl]-2H-isoindol-2-yl]-2,6-piperidinedione dihydrochloride

CAS Number

2520105-60-4

PubChem ID

155229258

InChI Key

GCOKMWGDIBQIRU-UHFFFAOYSA-N

SMILES

O=C1N(C2CCC(NC2=O)=O)CC3=CC(N4CCN(CC4)CC5CCNCC5)=CC=C13.Cl.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

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Background References

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Product Documents for Lenalidomide 5'-piperazine-4-methylpiperidine

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Lenalidomide 5'-piperazine-4-methylpiperidine

For research use only

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