ONO 8130

Tocris Bioscience | Catalog # 5406

EP1 receptor antagonist
Tocris Bioscience

Key Product Details

Description

EP1 receptor antagonist
View all Prostanoid Receptor Antagonists »

Product Description

ONO 8130 is an EP1 receptor antagonist. Exhibits analgesic effect in a mouse model of cystitis. Orally bioavailable.

Product Specifications for ONO 8130

Molecular Weight

500.63

Formula

C25H28N2O5S2

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

4-[[[2,3-Dihydro-6-[(2-methylpropyl)[(4-methyl-2-thiazolyl)sulfonyl]amino]-1H-indene-5yl]oxy]methyl]benzoic acid

CAS Number

459841-96-4

PubChem ID

9827317

InChI Key

IOXMDBQCUCDLAF-UHFFFAOYSA-N

SMILES

CC(C)CN(S(C3=NC(C)=CS3)(=O)=O)C1=C(OCC4=CC=C(C(O)=O)C=C4)C=C(CCC2)C2=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 50.06 100
Ethanol 10.01 20

Preparing Stock Solutions for ONO 8130

The following data is based on the product molecular weight 500.63.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.00 mL 9.99 mL 19.97 mL
5 mM 0.40 mL 2.00 mL 3.99 mL
10 mM 0.20 mL 1.00 mL 2.00 mL
50 mM 0.04 mL 0.20 mL 0.40 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 4 publications citing the usage of this product.

Product Documents for ONO 8130

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for ONO 8130

For research use only

Customer Reviews for ONO 8130 (1)

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  • ONO 8130
    Name: Melanie Ikeh
    Verified Customer | Posted 05/31/2017

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