TCS 2510

Tocris Bioscience | Catalog # 4069

Selective EP4 agonist
Tocris Bioscience

Key Product Details

Description

Selective EP4 agonist
View all Prostanoid Receptor Agonists »

Product Description

TCS 2510 is a highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM). Displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM.

Product Specifications for TCS 2510

Molecular Weight

383.49

Formula

C21H29N5O2

Storage

Store at -20°C

Purity

≥98% (HPLC)

Chemical Name

(5R)-5-[(3S)-3-Hydroxy-4-phenyl-1-buten-1-yl]-1-[6-(2H-tetrazol-5-yl)hexyl]-2-pyrrolidinone

CAS Number

346673-06-1

PubChem ID

9864831

InChI Key

JWYPJSNXPZTEHL-VJKINUSGSA-N

SMILES

O=C1N(CCCCCCC2=NN=NN2)[C@@H](/C=C/[C@H](CC3=CC=CC=C3)O)CC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble in ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml)

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 10 publications citing the usage of this product.

  • Billot Discovery of a potent and selective agonist of the prostaglandin EP4 receptor. Bioorg.Med.Chem.Lett.

Product Documents for TCS 2510

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for TCS 2510

For research use only

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