4 results for "Adenosine A3 Receptor Antagonists" in 产品
Adenosine A3 Receptor Antagonists
The adenosine A3 receptor is a member of the adenosine receptor group of G-protein-coupled receptors that also includes A1, A2A and A2B. They display high expression levels in the testes and mast cells of rats, with low expression levels in the thyroid, liver, kidney, heart, intestine and most brain areas. Adenosine A3 receptors play a role in mast cell degranulation, coronary vasodilation and protection from reperfusion. The human A3 receptor gene is localized on chromosome 1 (1p21-p13).
Highly potent and selective hA3 antagonist
| Chemical Name: | N-[9-Chloro-2-(2-furanyl)[1,2,4]-triazolo[1,5-c]quinazolin-5-yl]benzene acetamide |
| Purity: | ≥98% |
Potent, highly selective hA3 receptor antagonist/inverse agonist
| Chemical Name: | (8R)-8-Ethyl-1,4,7,8-tetrahydro-4-methyl-2-(2,3,5-trichlorophenyl)-5H-imidazo[2,1-i]purin-5-one monohydrochloride |
| Purity: | ≥98% |
Potent and selective A3 adenosine receptor antagonist
| Chemical Name: | N-[4-(3,5-Dimethylphenyl)-5-(4-pyridinyl)-2-thiazolyl]-3-pyridinecarboxamide dihydrochloride |
| Purity: | ≥98% |
Potent and selective hA2B/A3 adenosine receptor fluorescent antagonist
| Purity: | ≥95% |
