7 results for "Nuclear Receptor Agonists" in 产品

Nuclear Receptor Agonists

High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic

Alternate Names: Sobetirome
Chemical Name: 2-[4-[[4-Hydroxy-3-(1-methylethyl)phenyl]methyl]-3,5-dimethylphenoxy]acetic acid
Purity: ≥98%
High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic
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Selective Rev-Erbα agonist

Alternate Names: SR 6452
Chemical Name: 1,1-Dimethylethyl-N-[(4-chlorophenyl)methyl]-N-[(5-nitro-2-thienyl)methyl])glycinate
Purity: ≥98%
Selective Rev-Erbα agonist
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High affinity Nur77 agonist

Chemical Name: Ethyl 3,5-dihydroxy-2-(1-oxooctyl)-benzeneacetate
Purity: ≥98%
High affinity Nur77 agonist
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Rev-Erbα/β agonist

Chemical Name: Ethyl 3-[[[(4-chlorophenyl)methyl][(5-nitro-2-thienyl)methyl]amino]methyl]-1-pyrrolidinecarboxylate
Purity: ≥98%
Rev-Erbα/β agonist
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T cell-specific RORγ (RORγt) agonist

Chemical Name: 2-Chloro-N-[4-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenyl]benzamide
Purity: ≥98%
T cell-specific RORγ (RORγt) agonist
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Selective Rev-Erbα/β agonist; anxiolytic

Chemical Name: [3-[[4-(1,1-Dimethylethoxy)phenoxy]methyl]-3,4-dihydro-2(1H)-isoquinolinyl]-1-naphthalenylmethanone
Purity: ≥98%
Selective Rev-Erbα/β agonist; anxiolytic
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Nurr1 activator; inhibits NF-κB-dependent gene expression

Chemical Name: 3,3'-[(4-Chlorophenyl)methylene]bis[1H-indole]
Purity: ≥98%
Nurr1 activator; inhibits NF-κB-dependent gene expression
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