7 results for "transcriptional-cyclin-dependent-kinase-inhibitors&view=expanded" in 产品

Cdk8 inhibitor

Chemical Name: 4-[(2-Phenylethyl)amino]-6-quinazolinecarbonitrile hydrochloride
Purity: ≥98%
Cdk8 inhibitor
Loading...

Selective cdk7 inhibitor

Chemical Name: N5-(6-Aminohexyl)-3-(1-methylethyl)-N7-(phenylmethyl)pyrazolo[1,5-a]pyrimidine-5,7-diamine dihydrochloride
Purity: ≥98%
Selective cdk7 inhibitor
Loading...

Potent and selective CDK8 and CDK19 inhibitor; maintains pluripotency of mouse PSCs in culture

Chemical Name: N-Propyl-3-(4-pyridinyl)imidazo[1,2-b]pyridazin-6-amine
Purity: ≥98%
Potent and selective CDK8 and CDK19 inhibitor; maintains pluripotency of mouse PSCs in culture
Loading...

Potent and selective CDK7 inhibitor; induces cell cycle arrest

Chemical Name: N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[[4-[(1-oxo-2-propen-1-yl)amino]benzoyl]amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide
Purity: ≥95%
Potent and selective CDK7 inhibitor; induces cell cycle arrest
Loading...

Potent and selective ATP-competitive CDK9 inhibitor

Chemical Name: 4-[[[5'-Chloro-2'-[[trans-4-[[(1R)-2-methoxy-1-methylethyl]amino]cyclohexyl]amino][2,4'-bipyridin]-6-yl]amino]methyl]tetrahydro-2H-pyran-4-carbonitrile
Purity: ≥97%
Potent and selective ATP-competitive CDK9 inhibitor
Loading...

Potent and selective Cdk9 Degrader (PROTAC®)

Chemical Name: N-(5-(((5-(tert-Butyl)oxazol-2-yl)methyl)thio)thiazol-2-yl)-1-(14-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)-2-oxo-6,9,12-trioxa-3-azatetradecyl)piperidine-4-carboxamide
Purity: ≥98%
Application of THAL SNS 032 in MOLT-4 cells
(2)
Loading...

Molecular glue; induces degradation of CCNK and CDK12

Chemical Name: 6,7-Dihydro-N-(5-methyl-2-thiazolyl)-5H-indeno[5,6-b]furan-3-acetamide
Purity: ≥98%
Molecular glue; induces degradation of CCNK and CDK12
Loading...
Results Per Page
5 10 25 50
  • / 1