5 results for "TREK 1 Small Molecules and Peptides" in 产品
TREK 1 Small Molecules and Peptides
A potassium channel called TREK1 may represent a new target for antidepressant drugs, according to research published in the September issue of Nature Neuroscience. The channel may exert its effects through a signaling pathway in the brain that is different than what is normally targeted by most conventional antidepressants, which are thought to work by increasing the level of the neurotransmitter serotonin in the brain. Michel Lazdunski and colleagues studied mice lacking the gene for the ...
Selective K2P2.1 (TREK-1) and K2P10.1 (TREK-2) activator
| Chemical Name: | N-[(2,4-Dichlorophenyl)methyl]-4-[(methylsulfonyl)amino]benzamide |
| Purity: | ≥98% |
Potent K2P2.1 (TREK-1) channel blocker
| Purity: | ≥95% |
K2P2.1 (TREK-1) and K2P10.1 (TREK-2) channel activator
| Chemical Name: | 4,4'-[[2,2,2-Trifluoro-1-(trifluoromethyl)ethylidene]bis(4,1-phenyleneoxy)]bis[benzenamine] |
| Purity: | ≥99% |
Potent inhibitor of TREK-1 channels
| Purity: | ≥95% |
KV11.1 (hERG) channel blocker; inhibits rapid delayed rectifier K+ current (IKr)
| Alternate Names: | Tikosyn,UK 68798 |
| Chemical Name: | 1-(4-Methanesulphonamidophenoxy)-2-[N-(4-methanesulphonamidophenethyl)-N-methylamino]ethane |
| Purity: | ≥98% |
