14 results for "vasopressin-receptor-peptides&view=expanded" in 产品

Antidiuretic hormone

Alternate Names: AVP
Purity: ≥95%
Antidiuretic hormone
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Synthetic vasopressin analog; V1B and V2 agonist

Purity: ≥95%
Synthetic vasopressin analog; V1B and V2 agonist
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Selective vasopressin V1A antagonist

Purity: ≥95%
Selective vasopressin V1A antagonist
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Selective, orally active vasopressin V1A receptor antagonist

Alternate Names: Relcovaptan
Chemical Name: (2S)-1-[[(2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-[(3,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-hydroxy-1H-indol-2-yl]carbonyl]-2-pyrrolidinecarboxamide
Purity: ≥98%
Selective, orally active vasopressin V1A receptor antagonist
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Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active

Alternate Names: OPC-41061
Chemical Name: N-[4-[(7-Chloro-2,3,4,5-tetrahydro-5-hydroxy-1H-1-benzazepin-1-yl)carbonyl]-3-methylphenyl]-2-methylbenzamide
Purity: ≥98%
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active
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Potent and selective vasopressin V1B antagonist

Alternate Names: Nelivaptan
Chemical Name: (2S,4R)-1-[(3R)-5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-2,3-dihydro-3-(2-methoxyphenyl)-2-oxo-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidinecarboxamide
Purity: ≥98%
Potent and selective vasopressin V1B antagonist
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Reactivity: Human
Source: E. coli
Applications: AC
V1b Vasopressin R/AVPR1B Recombinant Protein Antigen
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Orally active vasopressin V1 antagonist

Chemical Name: N-[3-[4-[[4-(3,4-Dihydro-2-oxo-1(2H)quinolinyl)-1-piperidinyl]carbonyl]phenoxy]propyl]-acetamide
Purity: ≥98%
Orally active vasopressin V1 antagonist
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Potent and selective V1B receptor antagonist; orally bioavailable

Chemical Name: 2-(3-Chloro-4-fluorophenyl)-N-(1-methylethyl)-6-[3-(4-morpholinyl)propoxy]-4-oxo-pyrido[2,3-d]pyrimidine-3(4H)-acetamide hydrochloride
Purity: ≥98%
Potent and selective V1B receptor antagonist; orally bioavailable
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Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist

Chemical Name: (2S)-N-[[4-[(4,10-Dihydro-1-methylpyrazolo[3,4-b][1,5]benzodiazepin-5(1H)-yl)carbonyl]-2-methylphenyl]methyl]-2-[(hexahydro-4-methyl-1H-1,4-diazepin-1-yl)thioxomethyl]-1-pyrrolidinecarboxamide
Purity: ≥97%
Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist
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