4-PPBP maleate

Key Product Details

Product Description

4-PPBP maleate is a σ ligand and selective non-competitive antagonist at recombinant NR1a/2B NMDA receptors expressed in Xenopus oocytes.

Product Specifications for 4-PPBP maleate

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for 4-PPBP maleate

The following data is based on the product molecular weight 409.52.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.25 mM	9.77 mL	48.84 mL	97.68 mL
1.25 mM	1.95 mL	9.77 mL	19.54 mL
2.5 mM	0.98 mL	4.88 mL	9.77 mL
12.5 mM	0.20 mL	0.98 mL	1.95 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Whittemore Antagonism of N-MthD.-aspartate receptors by σ site ligands: potency, subtype-selectivity and mechanisms of inhibition. J.Pharmacol.Exp.Ther. 1997 PMID: 9223571
• Glennon Novel 1-phenylpiperazine and 4-phenylpiperidine derivatives as high affinity σ ligands. J.Med.Chem. 1991 PMID: 1662725

Product Documents for 4-PPBP maleate