Widely used H2
histamine antagonist which has more recently been described as an inverse agonist. Also a potent I1
imidazoline binding site ligand.
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All Tocris products are intended for laboratory research use only.
Distribution, properties and functional characteristics of three classes of histamine receptor.
The imidazoline I1 receptor agonist, moxonidine, inhibits insulin secretion from isolated rat islets of langerhans.
Tsoli et al.
Inverse agonism of histamine H2 antagonists accounts for upregulation of spontaneously active receptors.
Smit et al.
A second generation of centrally acting antihypertensive agents act on putative I1-imidazoline receptors.
Ernsberger et al.
The citations listed below are publications that use Tocris products. Selected citations for Cimetidine include:
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