Chemical Name: 17-(Cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α,α-dimethyl-6,14-ethenomorphinan-7-methanol
Biological ActivityDiprenorphine is a non-selective opioid receptor antagonist (Ki values are 0.017, 0.072 and 0.23 nM for κ-, μ- and δ-opioid receptors).
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Classification of opioid receptors.
Paterson et al.
Pharmacological characterization of the cloned κ-, δ-, and μ-opioid receptors.
Raynor et al.
The effect of the nonselective opioid antagonist diprenorphine vasopressin secretion in the rat.
Iwasaki et al.
Citation for Diprenorphine
The citations listed below are publications that use Tocris products. Selected citations for Diprenorphine include:
1 Citation: Showing 1 - 1
Separating myoblast differentiation from muscle cell fusion using IGF-I and the p38 MAP kinase inhibitor SB202190.
Authors: Gardner Et al.
Am J Physiol Cell Physiol 2015;309:C491
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Diprenorphine was use to displace radiolabeled-diprenorphine in an homologous radiobinding assay.