Catalog Number: 2965
Chemical Name: 17-(Cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α,α-dimethyl-6,14-ethenomorphinan-7-methanol
Biological Activity
Non-selective opioid receptor antagonist (Ki values are 0.017, 0.072 and 0.23 nM for κ-, μ- and δ-opioid receptors).
Technical Data
  • M.Wt:
    425.56
  • Formula:
    C26H35NO4
  • Solubility:
    Soluble to 20 mM in DMSO and to 25 mM in ethanol
  • Purity:
    >99%
  • Storage:
    Store at RT
  • CAS No:
    14357-78-9
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Classification of opioid receptors.
    Paterson et al.
    Br.Med.Bull., 1983;39:31
  2. Pharmacological characterization of the cloned κ-, δ-, and μ-opioid receptors.
    Raynor et al.
    Mol.Pharmacol., 1994;45:330
  3. The effect of the nonselective opioid antagonist diprenorphine vasopressin secretion in the rat.
    Iwasaki et al.
    Endocrinology, 1994;134:48

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