Potent and selective monoacylglycerol lipase (MAGL) inhibitor (IC50
= 3.7 nM). Displays >1000-fold selectivity for MAGL over fatty acid amide hydrolase (IC50
= 20.6 μM). Analog of JZL 195
(Cat. No. 4715).
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Highly selective inhibitors of monoacylglycerol lipase bearing a reactive group that is bioisosteric with endocannabinoid substrates.
Chang et al.