Antagonist at 5-HT1
with activity at 5-HT1D
. Has moderate affinity for 5-HT6
and high affinity for 5-HT7
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Effects of various serotonin receptor subtype selective antagonists alone and on m-chlorophenylpiperazine-induced neuroendocrine changes in rats.
Aulakh et al.
Pharmacological characterization of serotonin receptor subtypes involved in vasopressin and plasma renin activity responses to serotonin agonists.
Bagdy et al.
Agonist activity of sumatriptan and metergoline at the human 5-HT1Dβ receptor in the action of sumatriptan.
Miller et al.
The citations listed below are publications that use Tocris products. Selected citations for Metergoline include:
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