Potent and highly selective antagonist for the human adenosine A3
values are 2.69 nM at hA3
, and > 100 μ
M at rat A1
and rat A2A
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Sold with the permission of the NIH, US Patent 60/029,855
New potent and selective human adenosine A3 receptor antagonists.
Baraldi and Borea
Structure-activity relationships and molecular modeling of 3,5-diacyl-2,4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists.
Li et al.
The citations listed below are publications that use Tocris products. Selected citations for MRS 1334 include:
Showing Results 1 - 6 of 6