High affinity BRPF inhibitor (Kd
values are 40, 210 and 943 nM for BRPF1B, 2 and 3, respectively). Also exhibits modest activity at BRD9 (Kd
= 1130 nM). Exhibits selectivity for BRPF over 44 other bromodomains. Orally bioavailable.
Store at -20°C
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.