PHP 501 trifluoroacetate

Catalog # Availability Size / Price Qty
4466/10
4466/50
PHP 501 trifluoroacetate | CAS No. 1781880-44-1 | GABA-A Receptor Antagonists
1 Image
Description: Potent GABAA antagonist

Chemical Name: 4-(5-[1,1'-Biphenyl]-3-yl-1-hydroxy-1H-pyrazol-4-yl)piperidine trifluoroacetate

Purity: ≥98%

Product Details
Citations (2)
Supplemental Products
Reviews

Biological Activity

Potent GABAA antagonist (Ki = 0.0028 μM at rat GABAA receptors; IC50 = 0.024 μM at human α1β2γ2 GABAA-expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.

Technical Data

M.Wt:
433.42
Formula:
C20H21N3O.CF3CO2H
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1781880-44-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

Citations for PHP 501 trifluoroacetate

The citations listed below are publications that use Tocris products. Selected citations for PHP 501 trifluoroacetate include:

2 Citations: Showing 1 - 2

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

VersaClone cDNA Plasmids

Reviews for PHP 501 trifluoroacetate

There are currently no reviews for this product. Be the first to review PHP 501 trifluoroacetate and earn rewards!

Have you used PHP 501 trifluoroacetate?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.