= 0.0028 μ
M at rat GABAA
= 0.024 μ
M at human α1β2γ2
-expressing tsA201 cells). Displays no inhibitory activity at hGAT-1, hGAT-2, hGAT-3 or hBGT-1 GABA transporters.
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All Tocris products are intended for laboratory research use only.
Novel 4-(piperidin-4-yl)-1-hydroxypyrazoles as gamma-aminobutyric acid(A) receptor ligands: synthesis, pharmacology, and structure-activity relationships.
Møller et al.
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