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Pimozide

Catalog #: 0937 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
0937/100
Pimozide | CAS No. 2062-78-4 | Non-selective Dopamine Receptor Antagonists
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Description: D2-like antagonist; also high affinity 5-HT7 antagonist

Chemical Name: 1-[1-[4,4-Bis(4-fluorophenyl)butyl]-4-piperidinyl]-1,3-dihydro-2H-benzimidazol-2-one

Purity: ≥98%

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Biological Activity

Pimozide is a dopamine D2-receptor antagonist and antipsychotic which binds with very high affinity to the cloned rat 5-HT7 receptor (Ki = 0.5 nM).

Technical Data

M.Wt:
461.55
Formula:
C28H29F2N3O
Solubility:
Soluble to 20 mM in DMSO
Purity:
≥98%
Storage:
Store at RT
CAS No:
2062-78-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Complete Your Experiment

Human Dopamine D2 R/DRD2 (NP_000786) VersaClone cDNA
Cat # RDC0423

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⚠ WARNING: This product can expose you to chemicals including Pimozide, which is known to the State of California to cause reproductive toxicity with developmental effects. For more information, go to www.P65Warnings.ca.gov

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VersaClone cDNA Plasmids

Human Dopamine D2 R/DRD2 (NP_000786) VersaClone cDNA

RDC0423

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