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Spiroxatrine

Catalog #: 0631
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0631/50
Spiroxatrine | CAS No. 1054-88-2 | Adrenergic alpha-2 Receptor Antagonists
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Description: Potent α2C antagonist

Chemical Name: 8-[(2,3-Dihydro-1,4-benzodioxin-2-yl)methyl]-1-phenyl-1,3,8-triazaspiro[4,5]decan-4-one

Product Details
Citations (1)
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Biological Activity

Spiroxatrine is a 5-HT1A antagonist. More active and selective than spiperone. Also a very potent α2C adrenergic receptor antagonist.

Technical Data

M.Wt:
379.46
Formula:
C22H25N3O3
Solubility:
Soluble to 10 mM in DMSO
Storage:
Store at RT
CAS No:
1054-88-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Complete Your Experiment

Human ADRA2C (NP_000674) VersaClone cDNA
Cat # RDC0258

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Citation for Spiroxatrine

The citations listed below are publications that use Tocris products. Selected citations for Spiroxatrine include:

1 Citation: Showing 1 - 1

  1. Alpha2-adrenoceptor subtypes involved in the regulation of catecholamine release from the adrenal medulla of mice.
    Authors: Moura Et al.
    Br J Pharmacol  2006;149:1049

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VersaClone cDNA Plasmids

Human ADRA2C (NP_000674) VersaClone cDNA

RDC0258

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