Home / Phosphodiesterase Inhibitors / TC-E 5005

TC-E 5005

Catalog #: 4572 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
4572/10
4572/50
TC-E 5005 | CAS No. 959705-64-7 | Phosphodiesterase Inhibitors
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Description: Potent and selective PDE10A inhibitor

Chemical Name: 2-Methoxy-6,7-dimethyl-9-propyl-imidazo[1,5-a]pyrido[3,2-e]pyrazine

Purity: ≥99%

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Biological Activity

TC-E 5005 is a potent and selective PDE10A inhibitor (IC50 values are 7.28, 239, 779, 919, 3100 and 3700 nM at PDE10A, 2A, 11A, 5A, 7B and 3A respectively and >5000 nM at PDE1B, 4A, 6, 8A and 9A). Reverses MK 801-induced hyperactivity in vivo.

Technical Data

M.Wt:
270.33
Formula:
C15H18N4O
Solubility:
Soluble to 100 mM in 1eq. HCl and to 100 mM in ethanol
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
959705-64-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Product Datasheets

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