YM 202074 sesquifumarate

Catalog # Availability Size / Price Qty
3413/5
3413/25
YM 202074 sesquifumarate | CAS No. 299900-84-8 | Group I mGluR Antagonists
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Description: High affinity, selective mGlu1 antagonist

Chemical Name: N-Cyclohexyl-6-[[N-(2-methoxyethyl)-N-methylamino]methyl]-N-methylthiazolo[3,2-a]benzoimidazole-2-carboxamide sesquifumarate

Purity: ≥99%

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Biological Activity

High affinity, selective metabotropic glutamate receptor type 1 (mGlu1) antagonist. Binds an allosteric site of the rat mGlu1 receptor with a Ki of 4.8 nM. Inhibits mGlu1-mediated inositol phosphates production (IC50 = 8.6 nM in rat cerebellar granule cells). Neuroprotective in vivo.

Technical Data

M.Wt:
588.67
Formula:
C22H30N4O2S.1.5C4H4O4
Solubility:
Soluble to 20 mM in water and to 100 mM in DMSO
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
299900-84-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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