1 result for "Non-selective Endothelin Receptor Antagonists" in Products

Non-selective Endothelin Receptor Antagonists

EDNRA and EDNRB (endothelin A and B receptors, respectively) are members of the rhodopsin-like 7-transmembrane receptor family. EDNRA binds endothelins ET-1 and ET-2 preferentially, and is expressed on vascular smooth muscle where it mediates vasoconstriction. EDNRB binds all three endothelin forms equally, and is expressed on endothelial cells whe...

Show More

High affinity dual ETA and ETB receptor antagonist;orally bioavailable

Alternate Names: Ro 47-0203
Chemical Name: 4-(1,1-Dimethylethyl)-N-[6-(2-hydroxyethoxy)-5-(2-methoxyphenoxy)[2,2'-bipyrimidin]-4-yl]benzenesulfonamide
Purity: ≥98%
High affinity dual ETA and ETB receptor antagonist;orally bioavailable
Loading...
Results Per Page
5 10 25 50
  • / 1