2 results for "PAK4 Small Molecules and Peptides" in Products

PAK4 Small Molecules and Peptides

PAK (p21-activated kinases) are a family of serine/threonine kinases within the STE ser/thr protein kinase superfamily that play roles in various oncogenic signaling pathways. Cytoskeletal remodeling, motility, proliferation, and aberrant response to apoptosis and mitosis signals are among oncogenic cell functions coordinated by PAK family members....

Show More

Potent PAK4 inhibitor; orally available

Chemical Name: N-[(1S)-2-(Dimethylamino)-1-phenylethyl]-4,6-dihydro-6,6-dimethyl-3-[(2-methylthieno[3,2-d]pyrimidin-4-yl)amino]pyrrolo[3,4-c]pyrazole-5(1H)-carboxamide dihydrochloride
Purity: ≥98%
Potent PAK4 inhibitor; orally available
Loading...

Potent PAK inhibitor; brain penetrant and orally bioavailable

Chemical Name: 6-(2,4-Dichlorophenyl)-8-ethyl-2-[[3-fluoro-4-(1-piperazinyl)phenyl]amino]pyrido[2,3-d]pyrimidin-7(8H)-one
Purity: ≥98%
Potent PAK inhibitor; brain penetrant and orally bioavailable
Loading...
Results Per Page
5 10 25 50
  • / 1