PSB 0788

Key Product Details

Product Description

PSB 0788 is a potent and selective adenosine A_2B receptor antagonist (IC₅₀ = 3.64 nM at human A_2B receptors). Displays > 100-fold selectivity over hA₁, hA_2A and hA₃ receptors.

Product Specifications for PSB 0788

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for PSB 0788

The following data is based on the product molecular weight 543.04.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	1.84 mL	9.21 mL	18.41 mL
5 mM	0.37 mL	1.84 mL	3.68 mL
10 mM	0.18 mL	0.92 mL	1.84 mL
50 mM	0.04 mL	0.18 mL	0.37 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 6 publications citing the usage of this product.

• Borrmann 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity. J.Med.Chem. 2009 PMID: 19569717

Product Documents for PSB 0788