6 results for "Adenosine A2b Receptor Antagonists" in 产品
Adenosine A2b Receptor Antagonists
Adenosine A2B receptors are members of the adenosine receptor group of G-protein-coupled receptors that also includes A1, A2A and A3. A2B receptors display high expression levels in the cecum, colon and bladder, with lower levels found in the lung, blood vessels, eye, median eminence and mast cells. A2B receptors play a role in the relaxation of smooth muscle in the vasculature and intestines, inhibit monocyte and macrophage function and stimulate mast cell mediator release. The human A2B ...
Selective A2B antagonist
| Chemical Name: | N-(4-Cyanophenyl)-2-[4-(2,3,6,7-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]-acetamide |
| Purity: | ≥98% |
Selective human A2B antagonist; water-soluble
| Chemical Name: | 4-(2,3,6,7-Tetrahydro-2,6-dioxo-1-propyl-1H-purin-8-yl)-benzenesulfonic acid |
| Purity: | ≥98% |
Highly selective A2B antagonist
| Chemical Name: | 8-[4-[4-(4-Chlorophenzyl)piperazide-1-sulfonyl)phenyl]]-1-propylxanthine |
| Purity: | ≥98% |
Selective A2B antagonist
| Chemical Name: | 8-[4-[4-(4-Chlorobenzyl)piperazide-1-sulfonyl)phenyl]]-1-propylxanthine |
| Purity: | ≥98% |
Selective A2B antagonist
| Alternate Names: | CVT 6883 |
| Chemical Name: | 3-Ethyl-3,9-dihydro-1-propyl-8-[1-[[3-(trifluoromethyl)phenyl]methyl]-1H-pyrazol-4-yl]-1H-purine-2,6-dione |
| Purity: | ≥98% |
Potent and selective hA2B/A3 adenosine receptor fluorescent antagonist
| Purity: | ≥95% |