5 results for "Melanocortin Receptor Agonists" in 产品

Melanocortin Receptor Agonists

Melanocortin receptors are activated by members of the melanocortin family: α-, β- and γ-melanocyte stimulating hormone (MSH) and adrenocorticotropic hormone (ACTH). Endogenous antagonists include agouti and agouti-related protein (AgRP). The melanocortin receptors are G-protein-coupled and 5 subtypes exist, MC1-5. The melanocortins are involved in a wide range of physiological functions, including pigmentation, energy homeostasis, inflammation, immunomodulation, steroidogenesis and temperature control.

Endogenous melanocortin receptor agonist

Alternate Names: α-Melanotropin,α-Melanocyte-stimulating hormone
Purity: ≥95%
Endogenous melanocortin receptor agonist
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Melanocortin receptor agonist

Alternate Names: Melanotan I,MT-I,NDP-α-MSH
Purity: ≥95%
Melanocortin receptor agonist
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Potent endogenous MC2 agonist

Alternate Names: Adrenocorticotropic hormone (1-39)
Purity: ≥95%
Potent endogenous MC2 agonist
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Potent and selective MC4 receptor agonist

Chemical Name: N-[(1R)-1-[(4-Chlorophenyl)methyl]-2-[4-cyclohexyl-4-(1H-1,2,4-trazol-1-ylmethyl)-1-piperidinyl]-2-oxoethyl]-1,2,3,4-tetrahydro-3-isoquinolinecarboxamide
Purity: ≥95%
Potent and selective MC4 receptor agonist
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High affinity melanocortin receptor agonist

Alternate Names: MT-II
Purity: ≥95%
High affinity melanocortin receptor agonist
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