9 results for "Nicotinic (a4b2) Receptor Agonists Small Molecules and Peptides" in 产品

Nicotinic (a4b2) Receptor Agonists Small Molecules and Peptides

Nicotinic α4β2 receptors have high affinity for nicotine and account for >90% of [3H]-nicotine binding to brain tissues. A stoichiometry of (α4)2(β2)3 has been proposed, generating two agonist binding sites consistent with the model of the muscle nAChR.

Manipulation of the stoichiometry of α4β2 nAChRs expressed in Xenopus oocytes indicates that (α4)3(β2)2 nAChRs are also viable, displaying lower affinity for ACh and higher Ca2+ permeability; whether ...

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Prototypical nAChR agonist

Chemical Name: (S)-(-)-1-Methyl-2-(3-pyridyl)pyrrolidine (L-(+))-ditartrate salt
Purity: ≥99%
Prototypical nAChR agonist
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Selective α4β2 nAChR partial agonist; orally active

Chemical Name: 7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine tartrate
Purity: ≥99%
Selective α4β2 nAChR partial agonist; orally active
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Highly potent PSAM4-GlyR and PSAM4-5-HT3 chimeric ion channel agonist; brain-penetrant

Chemical Name: 1-Methyl-7,8,9,10-tetrahydro-1H-6,10-methanoazepino[4,5-g]quinoxalin-2(6H)-one hydrochloride
Purity: ≥98%
Highly potent PSAM4-GlyR and PSAM4-5-HT3 chimeric ion channel agonist; brain-penetrant
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Selective α4β2 nAChR agonist

Alternate Names: Metanicotine,TC-2403
Chemical Name: (E)-N-Methyl-4-(3-pyridinyl)-3-buten-1-amine oxalate
Purity: ≥99%
Selective α4β2 nAChR agonist
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Selective α4β2 nAChR partial agonist

Chemical Name: 4-(5-ethoxy-3-pyridinyl)-N-methyl-(3E)-3-buten-1-amine difumarate
Purity: ≥98%
Selective α4β2 nAChR partial agonist
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Potent α4β4, α4β2 and α7 nAChR agonist

Chemical Name: (1R,5S)-9-Bromo-1,2,3,4,5,6-hexahydro-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one
Purity: ≥98%
Potent α4β4, α4β2 and α7 nAChR agonist
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High affinity and selective α4β2 nAChR partial agonist

Chemical Name: 2-Methyl-3-[(2S)-pyrrolidinylmethoxy]pyridine dihydrochloride
Purity: ≥98%
High affinity and selective α4β2 nAChR partial agonist
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Potent positive allosteric modulator of α4β2 nAChRs; also inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs

Chemical Name: 3-(2-Chlorophenyl)-5-(5-methyl-1-(piperidin-4-yl)-1H-pyrazol-4-yl)isoxazole hydrochloride
Purity: ≥98%
Potent positive allosteric modulator of α4β2 nAChRs; also inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs
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Selective α4β2 nAChR agonist

Alternate Names: Tebanicline
Chemical Name: (R)-5-(Azetidin-2-ylmethoxy)-2-chloropyridine hydrochloride
Purity: ≥98%
Selective α4β2 nAChR agonist
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