3'-Fluorobenzylspiperone maleate

Key Product Details

Product Description

3'-Fluorobenzylspiperone maleate is a very potent and selective ligand for the D₂ receptor (K_i = 0.023 nM). Compared with spiperone, displays a 2.5-fold greater affinity at D₂ and a 12-fold lower affinity at 5-HT₂ receptors.

Product Specifications for 3'-Fluorobenzylspiperone maleate

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for 3'-Fluorobenzylspiperone maleate

The following data is based on the product molecular weight 619.67.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.25 mM	6.46 mL	32.28 mL	64.55 mL
1.25 mM	1.29 mL	6.46 mL	12.91 mL
2.5 mM	0.65 mL	3.23 mL	6.46 mL
12.5 mM	0.13 mL	0.65 mL	1.29 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Mach Effect of N-alkylation on the affinities of analogues of spiperone for DA D₂ and serotonin 5-HT₂ receptors. J.Med.Chem. 1992 PMID: 1531364

Product Documents for 3'-Fluorobenzylspiperone maleate