4F 4PP oxalate

Key Product Details

Product Description

4F 4PP oxalate is a selective 5-HT_2A antagonist with almost as high affinity (K_i = 5.3 nM) as Ketanserin (Cat. No. 0908) but with a much lower affinity for 5-HT_2C sites (K_i = 620 nM).

Product Specifications for 4F 4PP oxalate

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for 4F 4PP oxalate

The following data is based on the product molecular weight 429.49.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	2.33 mL	11.64 mL	23.28 mL
5 mM	0.47 mL	2.33 mL	4.66 mL
10 mM	0.23 mL	1.16 mL	2.33 mL
50 mM	0.05 mL	0.23 mL	0.47 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 6 publications citing the usage of this product.

• Herndon Ketanserin analogues - structure affinity relationships of 5HT₂ and 5HT_1C serotonin receptor binding. J.Med.Chem. 1992 PMID: 1479590
• Hagberg Stimulation of 5-HT_2A receptors on astrocytes in primary culture opens voltage-independent Ca²⁺ channels. Neurochem.Int. 1998 PMID: 9542727

Product Documents for 4F 4PP oxalate