Ketanserin tartrate

Tocris Bioscience | Catalog # 0908

Selective 5-HT2A antagonist. Also antagonist at 5-HT1D
Tocris Bioscience

Key Product Details

Description

Selective 5-HT2A antagonist. Also antagonist at 5-HT1D

Alternative Names

R 41 468
View all 5-HT2A Receptor Antagonists »

Product Description

Ketanserin tartrate is a selective 5-HT2A serotonin receptor antagonist; can also be used to discriminate between 5-HT1D and 5-HT1B receptor subtypes.

Product Specifications for Ketanserin tartrate

Molecular Weight

545.52

Formula

C22H22FN3O3.C4H6O6

Storage

Store at RT

Purity

≥97% (HPLC)

Chemical Name

3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4[1H,3H]-quinazolinedione (L)-tartrate

CAS Number

83846-83-7

PubChem ID

135348

InChI Key

KMTLTEVOQLMYRS-UHFFFAOYSA-N

SMILES

OC(C(O)C(O)=O)C(O)=O.FC1=CC=C(C=C1)C(=O)C1CCN(CCN2C(=O)NC3=CC=CC=C3C2=O)CC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 5.45 10

Preparing Stock Solutions for Ketanserin tartrate

The following data is based on the product molecular weight 545.52.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.33 mL 91.66 mL 183.31 mL
0.5 mM 3.67 mL 18.33 mL 36.66 mL
1 mM 1.83 mL 9.17 mL 18.33 mL
5 mM 0.37 mL 1.83 mL 3.67 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 69 publications citing the usage of this product.

Product Documents for Ketanserin tartrate

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Ketanserin tartrate

For research use only

Citations for Ketanserin tartrate

Customer Reviews for Ketanserin tartrate (2)

5 out of 5
2 Customer Ratings
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4 Stars
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1 Stars
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  • Ketanserin
    Name: Nora Digranes
    Species: Pig
    Verified Customer | Posted 05/14/2024
    Tocris was very helpful in providing information on how to solve to powder.
    As a 5HT2A antagonist in a porcine model
  • Antidepressantsby Cholecystokinin Neurons of the Dentate Gyrus
    Name: Anonymous
    Species: Mouse
    Assay Type: In Vivo
    Verified Customer | Posted 02/03/2020
    20mM ketanserin
    Ketanserin tartrate 0908

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