Chemical Name:Ethyl 2-[[3,4-dihydro-4-oxo-3-[3-(1-pyrrolidinyl)propyl]benzothieno[3,2-d]pyrimidin-2-yl]thio]acetate
Biological Activity ALDH1A1 inhibitor (IC50 = 4.6 μM; Ki = 300 nM). Exhibits selectivity for ALDH1A1 over eight other ALDH isoforms. Disrupts spheroid formation and reduces cell viability of ovarian cancer cells in vitro.
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Store at +4°C
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