endothelin receptor agonist (IC50
values are 0.33 and 2200 nM for displacing [125
I]-ET-1 from ETB
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Endothelin and structurally related analogs distinguish between endothelin receptor subtypes.
Panek et al.
Different distribution of endothelin receptor subtypes in pulmonary tissues revealed by the novel selective ligands BQ-123 and [Ala1,3,11,15]ET1.
Nakamichi et al.