Potent and selective 5-HT2A
receptor antagonist (Ki
values are 0.13, 4.55, 40, 62 and 1570 nM at 5-HT2A
respectively). Centrally active following systemic administration in vivo
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All Tocris products are intended for laboratory research use only.
Synthesis and in vitro affinities of various MDL 100907 derivatives as potential 18F-radioligands for 5-HT2A receptor imaging with PET.
Herth et al.
Stimulation of corticosterone and β-endorphin secretion in the rat by selective 5-HT receptor subtype activation.
Koenig et al.
Evidence that 5-HT2C receptor antagonists are anxiolytic in the rat Geller-Seifter model of anxiety.
Kennett et al.
Involvement of 5-HT2 receptors in the LSD- and L-5-HTP-induced suppression of lordotic behavior in the female rat.
J.Neural Transm., 1985;61:65
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