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Bay 59-3074

Catalog #: 2500
2 Citations Datasheet / COA / SDS

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2500 has been discontinued.
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Bay 59-3074 | CAS No. 406205-74-1 | Non-selective Cannabinoid Receptor Agonists
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Description: CB1/CB2 receptor partial agonist

Chemical Name: 3-[2-Cyano-3-(trifluoromethyl)phenoxy]phenyl 4,4,4-trifluoro-1-butanesulfonic acid ester

Purity: ≥99%

Product Details
Citations (2)
Reviews
Biological Activity Technical Data Additional Information Background Product Datasheets Calculators

Biological Activity

Bay 59-3074 is a novel CB1/CB2 receptor partial agonist (Ki values are 48.3 and 45.5 nM at human CB1 and CB2 receptors respectively). Orally active CB1 agonist in vivo. Displays anti-hyperalgesic and antiallodynic properties in rat models of chronic neuropathic and inflammatory pain.

Technical Data

M.Wt:
453.35
Formula:
C18H13F6NO4S
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
406205-74-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold for research purposes under agreement from Bayer

Product Datasheets

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Citations for Bay 59-3074

The citations listed below are publications that use Tocris products. Selected citations for Bay 59-3074 include:

2 Citations: Showing 1 - 2

  1. Pharmacological characterization of the P2 receptors profile in the podocytes of the freshly isolated rat glomeruli.
    Authors: Ilatovskaya Et al.
    Am J Physiol Cell Physiol  2013;305:C1050
  2. Characterizing cannabinoid CB2 receptor ligands using DiscoveRx PathHunter β-arrestin assay.
    Authors: McGuinness Et al.
    Biol Psychiatry  2009;14:49

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