Catalog Number: 4117
Chemical Name: N-Benzyl-N-(3-isobutoxy-2-pyrrolidin-1-yl-propyl)aniline hydrochloride
Biological Activity
Calcium channel blocker. Also inhibits Na+/Ca2+ exchange (NCX), sodium channels and cardiac sarcolemmal KATP channels; opens mitochondrial KATP channels. Antiarrhythmic and antihypertensive; acts as a calcium sensitizer.
Technical Data
  • M.Wt:
  • Formula:
  • Solubility:
    Soluble to 100 mM in DMSO
  • Purity:
  • Storage:
    Desiccate at RT
  • CAS No:
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Bepridil block of cardiac calcium and sodium channels.
    Yatani et al.
    J.Pharmacol.Exp.Ther., 1986;237:9
  2. Blocking effect of bepridil on Na+/ Ca2+ exchange current in gunea pig cardiac ventricular myocytes.
    Wantanabe and Kimura
    Jpn.J.Pharmacol., 2001;85:370
  3. Bepridil, an antiarrythmic drug, opens mitochondrial KATP channels, blocks sarcolemmal KATP channels, and confers cardioprotection.
    Sato et al.
    J.Pharmacol.Exp.Ther., 2006;316:182
  4. Pharmacology of bepridil.
    Gill et al.
    Am.J.Cardiol., 1992;69:11D

The citations listed below are publications that use Tocris products. Selected citations for Bepridil hydrochloride include:

1 Citations: Showing 1 - 1

  1. Intracellular and extracellular pH and Ca are bound to control mitosis in the early sea urchin embryo via ERK and MPF activities.
    Authors: Ciapa and Philippe
    PLoS One 2013;8:e66113

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