BI 01383298

Key Product Details

Product Description

BI 01383298 is a potent and selective inhibitor of human SLC13A5 (Na⁺/citrate cotransporter; IC₅₀ = 56 nM in HEK cells overexpressing hSLC13A5 and 24 nM in HepG2 cells with endogenous SLC13A5 expression). Displays >1000-fold selectivity over other family members.

Licensing Information

This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the BI01383298 probe summary on the SGC website.

Product Specifications for BI 01383298

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for BI 01383298

The following data is based on the product molecular weight 445.34.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.5 mM	4.49 mL	22.45 mL	44.91 mL
2.5 mM	0.90 mL	4.49 mL	8.98 mL
5 mM	0.45 mL	2.25 mL	4.49 mL
25 mM	0.09 mL	0.45 mL	0.90 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Peters Flipping a citrate switch on liver cancer cells. J.Biol.Chem. 2017 PMID: 28821606

Product Documents for BI 01383298