Selective neuromedin B receptor (NMB-R, BB1
) antagonist (Ki
values are 216 and 18,264 nM for BB1
receptors respectively). Displays no activity at a range of other receptors.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Discovery of a novel class of neuromedin B receptor antagonists, substituted somatostatin analogues.
Orbuch et al.
Pharmacological profiles of two bombesin analogues in cells transfected with human neuromedin B receptors.
Ryan et al.
Role of different bombesin receptor subtypes mediating contractile activity in cat upper gastrointestinal tract.
Milusheva et al.