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BMY 14802 hydrochloride

  ( 2 citations )    
Product Datasheet
Catalog Number:1440
Chemical Name:α-(4-Fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazinebutanol hydrochloride
Product Details
Citations (2)
Reviews
Biological Activity
Potent sigma receptor antagonist (IC50 = 112 nM) with modest to weak affinity for 5-HT1A and α1 receptors. Antipsychotic following oral administration and acts via indirect modulation of central dopaminergic systems.
Technical Data
  • M.Wt:
    384.86
  • Formula:
    C18H22F2N4O.HCl
  • Solubility:
    Soluble to 25 mM in water
  • Purity:
    >98
  • Storage:
    Desiccate at RT
  • CAS No:
    105565-55-7
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Additional Information
Licensing Caveats:
Sold with the permission of Bristol-Myers Squibb Company
Product Datasheets
SDS
COA view current batch
Citations:

The citations listed below are publications that use Tocris products. Selected citations for BMY 14802 hydrochloride include:

2 Citations: Showing 1 - 2
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  1. The effects of BMY-14802 against L-DOPA- and dopamine agonist-induced dyskinesia in the hemiparkinsonian rat.
    Authors: Bhide Et al.
    Psychopharmacology (Berl)  2013;227:533
  2. σ ligands, but not N-methyl-D-aspartate antagonists, reduce levodopa-induced dyskinesias.
    Authors: Paquette Et al.
    Reprod Biol Endocrinol  2008;19:111

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