Potent, selective ETB
receptor antagonist (IC50
= 1.2 nM for inhibition of ET-1 binding to human Girardi heart cells).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Biochemical and pharmacological profile of a potent and selective endothelin B-receptor antagonist, BQ-788.
Ishikawa et al.
International Union of Pharmacology. XXIX. Update on endothelin receptor nomenclature.
BQ-788, a selective endothelin ETB receptor antagonist.
Okada and Nishikibe
Cardiovasc.Drug Rev., 2002;20:53
The citations listed below are publications that use Tocris products. Selected citations for BQ 788 sodium salt include:
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