BRL 52537 hydrochloride

Key Product Details

Product Description

The most κ/μ-selective and among the most potent κ ligands known (25 times more potent than morphine in vivo).

Licensing Information

Sold with the permission of GlaxoSmithKline

Product Specifications for BRL 52537 hydrochloride

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for BRL 52537 hydrochloride

The following data is based on the product molecular weight 391.77.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

3 Recalculate

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.05 mM	51.05 mL	255.25 mL	510.50 mL
0.25 mM	10.21 mL	51.05 mL	102.10 mL
0.5 mM	5.11 mL	25.53 mL	51.05 mL
2.5 mM	1.02 mL	5.11 mL	10.21 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 5 publications citing the usage of this product.

• Vecchietti (2S)-1-(Arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective κ opioid analgesics. J.Med.Chem. 1991 PMID: 1846921

Product Documents for BRL 52537 hydrochloride