CGP 36216 hydrochloride

Key Product Details

Product Description

CGP 36216 hydrochloride is a selective GABA_B antagonist. Displays activity at presynaptic receptors; ineffective at GABA_B postsynaptic receptors.

Product Specifications for CGP 36216 hydrochloride

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for CGP 36216 hydrochloride

The following data is based on the product molecular weight 187.60.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	5.33 mL	26.65 mL	53.30 mL
5 mM	1.07 mL	5.33 mL	10.66 mL
10 mM	0.53 mL	2.67 mL	5.33 mL
50 mM	0.11 mL	0.53 mL	1.07 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 3 publications citing the usage of this product.

• Froestl Phosphinic acid analogues of GABA. 2. Selective, orally active GABA_B antagonists. J.Med.Chem. 1995 PMID: 7650685
• Ong CGP 36216 is a selective antagonist at GABA_B presynaptic receptors in rat brain. Eur.J.Pharmacol. 2001 PMID: 11274998

Product Documents for CGP 36216 hydrochloride