CID 1375606

Key Product Details

Product Description

CID 1375606 is a GPR27 agonist. Promotes recruitment of β-arrestin 2 to chimeric GPR27V₂ and wild-type GPR27 in a firefly luciferase complementation assay (pEC₅₀ values are 6.34 and 5.1, respectively).

Product Specifications for CID 1375606

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for CID 1375606

The following data is based on the product molecular weight 385.24.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
1 mM	2.60 mL	12.98 mL	25.96 mL
5 mM	0.52 mL	2.60 mL	5.19 mL
10 mM	0.26 mL	1.30 mL	2.60 mL
50 mM	0.05 mL	0.26 mL	0.52 mL

Calculators

Background References

References are publications that support the biological activity of the product.

• Dupuis Activation of the orphan G protein-coupled receptor GPR27 by surrogate ligands promotes β-arrestin 2 recruitment. Mol.Pharmacol. 2017 PMID: 28314853

Product Documents for CID 1375606