Deltarasin

Catalog # Availability Size / Price Qty
5424/10
Cat.No. 5424 - Deltarasin | C40H37N5O.3HCl | CAS No. 1440898-82-7
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Description: High affinity PDEδ-KRAS interaction inhibitor

Chemical Name: 2-[4-[(2S)-2-(2-Phenyl-1H-benzimidazol-1-yl)-2-(4-piperidinyl)ethoxy]phenyl]-1-(phenylmethyl)-1H-benzimidazole trihydrochloride

Product Details
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Biological Activity

High affinity PDEδ-KRAS interaction inhibitor (Kd = 41 nM); binds to PDEδ. Reduces proliferation and induces cell death of KRAS-dependent Panc-Tu-1 and Capan-1 pancreatic cancer cells. Attenuates tumor growth of Panc-Tu-1 xenografts in mice.

Technical Data

Formula:
C40H37N5O.3HCl
Solubility:
Soluble to 100 mM in water and to 100 mM in DMSO
Storage:
Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date.
CAS No:
1440898-82-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

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