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DV 7028 hydrochloride

Catalog #: 4480 Datasheet / COA / SDS

Discontinued Product

4480 has been discontinued.
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DV 7028 hydrochloride | CAS No. 133364-62-2 | 5-HT2A Receptor Antagonists
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Description: Selective 5-HT2A antagonist; antithrombotic

Chemical Name: 3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2H-pyrido[1,2-a]-1,3,5-triazine-2,4(3H)-dione hydrochloride

Purity: ≥99%

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Biological Activity

DV 7028 hydrochloride is a selective 5-HT2A receptor antagonist (Ki = 22 nM for at 5-HT2 receptors). Exhibits no affinity for 5-HT1A, 5-HT1B or 5-HT1D receptors. Inhibits collagen-induced serotonin secretion and platelet aggregation; displays no effect on serotonin uptake by platelets. Shown to inhibit arterial thrombus formation, but not venous thrombosis, in rat models.

Technical Data

M.Wt:
436.91
Formula:
C21H25FN4O3.HCl
Solubility:
Soluble to 10 mM in water with gentle warming and to 10 mM in DMSO with gentle warming
Purity:
≥99%
Storage:
Desiccate at RT
CAS No:
133364-62-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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