Home / mu Opioid Receptor Agonists / Endomorphin-1

Endomorphin-1

Catalog #: 1055
3 Citations Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
1055/5
Endomorphin-1
1 Image
Description: Potent and selective μ agonist

Purity: ≥95%

Product Details
Citations (3)
Supplemental Products
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Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

Endomorphin-1 is a endogenous peptide with an exceptionally high affinity (Ki = 360 pM) and selectivity for μ opioid receptors (4000- and 15000-fold preference over δ and κ respectively).

Technical Data

M.Wt:
610.67
Formula:
C34H38N6O5
Sequence:
YPWF

(Modification: Phe-4 = C-terminal amide)

Solubility:
Soluble to 0.60 mg/ml in water
Purity:
≥95%
Storage:
Store at -20°C
CAS No:
189388-22-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citations for Endomorphin-1

The citations listed below are publications that use Tocris products. Selected citations for Endomorphin-1 include:

3 Citations: Showing 1 - 3

  1. Pharmacogenomics of GPCR Drug Targets.
    Authors: Hauser Et al.
    Cell  2018;172:41
  2. Morphine-stimulated nitric oxide release in rabbit aqueous humor.
    Authors: Dortch-Carnes and Russell
    Am J Physiol Endocrinol Metab  2007;84:185
  3. RGSZ1 and GAIP regulate mu- but not delta-opioid receptors in mouse CNS: role in tachyphylaxis and acute tolerance.
    Authors: Garzón Et al.
    Neuropsychopharmacology  2004;29:1091

FAQs

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VersaClone cDNA Plasmids

Human mu Opioid R/OPRM1 (NP_000905) VersaClone cDNA

RDC0530

Rat mu Opioid R/OPRM1 (NP_037203) VersaClone cDNA

RDC0419

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