Chemical Name: 1,3,5-Trimethyl-2-[(4-methylphenyl)sulfonyl]benzene
Biological ActivityEPAC2 inhibitor. Inhibits cAMP binding to EPAC2 and cAMP mediated EPAC2 guanine nucleotide exchange factor (GEF) activity (IC50 = 0.4 μM).
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Tocris products are intended for laboratory research use only, unless stated otherwise.
Isoform-specific antagonists of exchange proteins directly activated by cAMP.
Tsalkova et al.
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