Flupirtine maleate

Catalog # Availability Size / Price Qty
2867/10
2867/50

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Flupirtine maleate | CAS No. 75507-68-5 | Non-selective/Other Potassium Channel Activators
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Description: KV7 channel activator; also GABAA modulator and indirect NMDA antagonist
Alternative Names: D 9998

Chemical Name: N-[2-Amino-6-[[4-fluorophenyl)methyl]amino]-3-pyridinyl]carbamic acid ethyl ester maleate

Purity: ≥98%

Product Details
Citations (2)
Reviews

Biological Activity

Flupirtine maleate is a non-opioid analgesic with muscle relaxant properties. Activates KV7 potassium channels, indirectly antagonizes NMDA receptors and modulates GABAA receptors. Exhibits neuroprotective actions in a model of cerebral ischemia in mice and reduces apoptosis and necrosis induced by noxious stimuli.

Technical Data

M.Wt:
420.4
Formula:
C15H17FN4O2.C4H4O4
Solubility:
Soluble to 100 mM in DMSO and to 10 mM in ethanol
Purity:
≥98%
Storage:
Desiccate at +4°C
CAS No:
75507-68-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for Flupirtine maleate

The citations listed below are publications that use Tocris products. Selected citations for Flupirtine maleate include:

2 Citations: Showing 1 - 2

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