Galnon

Tocris Bioscience | Catalog # 2085

Non-selective galanin receptor agonist
Tocris Bioscience
Discontinued Product
2085 has been discontinued. View all Galanin Receptor Agonists products.

Key Product Details

Description

Non-selective galanin receptor agonist
View all Galanin Receptor Agonists »

Product Description

Galnon is a novel non-peptide galanin GAL1 and GAL2 receptor agonist (Ki values are 11.7 and 34.1 μM respectively). Stimulates insulin release in isolated pancreatic islets from normal and diabetic rats. Systemically active in vivo; displays anticonvulsant activity following i.p. administration in mice. Central and peripheral administration also transiently inhibits food intake in rats and mice.

Product Specifications for Galnon

Molecular Weight

678.83

Formula

C40H46N4O6

Storage

Desiccate at -20°C

Chemical Name

3-Cyclohexyl-N-[(9H-fluoren-9-ylmethoxy)carbonyl]-L-alanyl-N-(4-methyl-2-oxo-2H-1-benzopyran-7-yl)-L-lysinamide

CAS Number

475115-35-6

PubChem ID

5311268

InChI Key

IKNOZZKXIDSTRN-PXLJZGITSA-N

SMILES

CC1=CC(=O)OC2=C1C=CC(NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC1CCCCC1)NC(=O)OCC1C3=CC=CC=C3C3=C1C=CC=C3)=C2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solubility Soluble to 67.88mg/ml in DMSO and to 16.97mg/ml in Ethanol with gentle warming

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 19 publications citing the usage of this product.

Product Documents for Galnon

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Galnon

For research use only

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